Reaction Details  Report a problem with these data
Target
Norepinephrine transporter
Ligand
BDBM50029150
Substrate
n/a
Ki
513±n/a nM
Comments
PDSP_976
Citation
 Shank, RP; Vaught, JL; Pelley, KA; Setler, PE; McComsey, DF; Maryanoff, BE McN-5652: a highly potent inhibitor of serotonin uptake. J Pharmacol Exp Ther 247:1032-8 (1988) [PubMed]
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM50029150
Synonyms:
3-(2-Piperidin-4-yl-ethyl)-1H-indole | CHEMBL276520 | Indalpine
Type:
Small organic molecule
Emp. Form.:
C15H20N2
Mol. Mass.:
228.3327
SMILES:
C(Cc1c[nH]c2ccccc12)C1CCNCC1
Structure:
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