Reaction Details  Report a problem with these data
Target
D1 dopamine receptor
Ligand
BDBM82247
Substrate
n/a
Ki
1.3±n/a nM
Comments
PDSP_1685
Citation
 Watts, VJ; Lawler, CP; Gilmore, JH; Southerland, SB; Nichols, DE; Mailman, RB Dopamine D1 receptors: efficacy of full (dihydrexidine) vs. partial (SKF38393) agonists in primates vs. rodents. Eur J Pharmacol 242:165-72 (1993) [PubMed]  Article
Target
Name:
D1 dopamine receptor
Synonyms:
D1 dopamine receptor | DOPAMINE D1 | DRD1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
8818.33
Organism:
Monkey
Description:
Q5I6B7
Residue:
78
Sequence:
VIMGVFVCCWLPFFILNCILPFCGSGETQPFCIDSITFDVFVWFGWANSSLNPIIYAFNADFRKAFSTLLGCYRLCPA
  
Inhibitor
Name:
BDBM82247
Synonyms:
8-Chloro-3-methyl-5-phenyl-2,3,4,5-tetrahydro-1H-benzo[d]azepin-7-ol(SCH 23390) | CAS_87134-87-0 | CHEMBL2158641 | CHEMBL62 | SCH 23388 | SCH 23390 | SCH 23390 (R-enantiomer) | SCH 23390,R(+)
Type:
Small organic molecule
Emp. Form.:
C17H18ClNO
Mol. Mass.:
287.784
SMILES:
CN1CCc2cc(Cl)c(O)cc2[C@H](C1)c1ccccc1 |r|
Structure:
Search PDB for entries with ligand similarity: