Reaction Details Report a problem with these data
Target
Alpha-2B adrenergic receptor
Ligand
BDBM50020192
Substrate
n/a
Ki
0.61±n/a nM
Comments
PDSP_1743
Citation
O'Rourke, MF; Blaxall, HS; Iversen, LJ; Bylund, DB Characterization of [3H]RX821002 binding to alpha-2 adrenergic receptor subtypes. J Pharmacol Exp Ther 268:1362-7 (1994) [PubMed]
More Info.:
Target
Name:
Alpha-2B adrenergic receptor
Synonyms:
ADA2B_DIDVI | ADRA2B | Alpha-2B adrenergic receptor | adrenergic Alpha2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
41875.91
Organism:
OPOSSUM
Description:
adrenergic Alpha2 0 OPOSSUM::O77715
Residue:
382
Sequence:
AIAAVITFLILFTIFGNALVILAVLTSRSLRAPQNLFLVSLAAADILVATLIIPFSLANELLGYWYFRHTWCEVYLALDVLFCTSSIVHLCAISLDRYWSVSRALEYNSKRTPRRIKGIILTVWLIAAFISLPPLIYKGDKGKKPGGRPQCKLNEEAWYILSSSIGSFFAPCLIMILVYLRIYLIAKRRNRQGPHGKQAPGDGDTGPSALGGTSTISKLPPSILPAVGEANGHSKPPGEREGGEQMGDPTSPSTPPNQSSVGPEDGSQKQEEEEEEEEEEEEECGPPAPPTSSSLQGTPNFQPSQGSQVLATLRGQVLLARGPASLGLQPWRRRTQMNREKRFTFVLAVVIGVFVLCWFPFFFSYSLGAICPQHCKVPHGLF