Reaction Details
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Target
Excitatory amino acid transporter 4
Ligand
BDBM50366648
Substrate
n/a
Meas. Tech.
ChEMBL_1735433 (CHEMBL4150969)
IC50
71±n/a nM
Citation
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More Info.:
Target
Name:
Excitatory amino acid transporter 4
Synonyms:
EAA4_RAT | Eaat4 | Excitatory amino acid transporter 4 | High-affinity neuronal glutamate transporter | Slc1a6 | Sodium-dependent glutamate/aspartate transporter | Solute carrier family 1 member 6
Type:
PROTEIN
Mol. Mass.:
60724.56
Organism:
Rattus norvegicus
Description:
ChEMBL_100180
Residue:
561
Sequence:
MSSHGNSLFLRESGAGGGCLQGLQDSLQQRALRTRLRLQTMTREHVRRFLRRNAFILLTVSAVIIGVSLAFALRPYQLTYRQIKYFSFPGELLMRMLQMLVLPLIVSSRVTGMASLDNKATGRMGMRAAVYYMVTTVIAVFIGILMVTIIHPGKGSKEGLHREGRIETVPTADAFMDLVRNMFPPNLVEACFKQFKTQYSTRVVTRTIVRTDNGSELGASISPPSSAENETSILENVTRALGTLQEVISFEETVPVPGSANGINALGLVVFSVAFGLVIGGMKHKGRVLRDFFDSLNEAIMRLVGIIIWYAPVGILFLIAGKILEMEDMAVLGGQLGMYTLTVIVGLFLHAGGVLPLIYFLVTHRNPFPFIGGILQALITAMGTSSSSATLPITFRCLEEGLGVDRRITRFVLPVGATVNMDGTALYEALAAIFIAQVNNYELNLGQITTISITATAASVGAAGIPQAGLVTMVIVLTSVGLPTEDITLIIAVDWFLDRLRTMTNVLGDSIGAAVIEHLSQRELELQEAELTLPSLGKPYKSLMAQAKGASRGRGGNESVM