Reaction Details
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Target
RAC-alpha serine/threonine-protein kinase
Ligand
BDBM50449751
Substrate
n/a
Meas. Tech.
ChEMBL_1740582 (CHEMBL4156332)
IC50
2600±n/a nM
Citation
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More Info.:
Target
Name:
RAC-alpha serine/threonine-protein kinase
Synonyms:
2.7.11.1 | AKT1_RAT | Akt1 | PKB | PKB alpha | Protein kinase B | Protein kinase B alpha | RAC-PK-alpha | RAC-alpha serine/threonine-protein kinase
Type:
PROTEIN
Mol. Mass.:
55728.72
Organism:
Rattus norvegicus
Description:
ChEMBL_102911
Residue:
480
Sequence:
MNDVAIVKEGWLHKRGEYIKTWRPRYFLLKNDGTFIGYKERPQDVEQRESPLNNFSVAQCQLMKTERPRPNTFIIRCLQWTTVIERTFHVETPEEREEWTTAIQTVADGLKRQEEETMDFRSGSPSDNSGAEEMEVALAKPKHRVTMNEFEYLKLLGKGTFGKVILVKEKATGRYYAMKILKKEVIVAKDEVAHTLTENRVLQNSRHPFLTALKYSFQTHDRLCFVMEYANGGELFFHLSRERVFSEDRARFYGAEIVSALDYLHSEKNVVYRDLKLENLMLDKDGHIKITDFGLCKEGIKDGATMKTFCGTPEYLAPEVLEDNDYGRAVDWWGLGVVMYEMMCGRLPFYNQDHEKLFELILMEEIRFPRTLGPEAKSLLSGLLKKDPTQRLGGGSEDAKEIMQHRFFANIVWQDVYEKKLSPPFKPQVTSETDTRYFDEEFTAQMITITPPDQDDSMECVDSERRPHFPQFSYSASGTA