Reaction Details Report a problem with these data
Target
Potassium voltage-gated channel subfamily A member 3
Ligand
BDBM50456969
Substrate
n/a
Meas. Tech.
ChEMBL_1758565 (CHEMBL4193573)
IC50
>10000±n/a nM
Citation
More Info.:
Target
Name:
Potassium voltage-gated channel subfamily A member 3
Synonyms:
KCNA3_RAT | Kcna3 | Potassium voltage-gated channel subfamily A member 3 | RCK3 | RGK5 | Voltage-gated potassium channel subunit Kv1.3 | Voltage-gated potassium channel subunit Kv3
Type:
PROTEIN
Mol. Mass.:
58414.47
Organism:
Rattus norvegicus
Description:
ChEMBL_100110
Residue:
525
Sequence:
MTVVPGDHLLEPEAAGGGGGDPPQGGCVSGGGCDRYEPLPPALPAAGEQDCCGERVVINISGLRFETQLKTLCQFPETLLGDPKRRMRYFDPLRNEYFFDRNRPSFDAILYYYQSGGRIRRPVNVPIDIFSEEIRFYQLGEEAMEKFREDEGFLREEERPLPRRDFQRQVWLLFEYPESSGPARGIAIVSVLVILISIVIFCLETLPEFRDEKDYPASPSQDVFEAANNSTSGASSGASSFSDPFFVVETLCIIWFSFELLVRFFACPSKATFSRNIMNLIDIVAIIPYFITLGTELAERQGNGQQAMSLAILRVIRLVRVFRIFKLSRHSKGLQILGQTLKASMRELGLLIFFLFIGVILFSSAVYFAEADDPSSGFNSIPDAFWWAVVTMTTVGYGDMHPVTIGGKIVGSLCAIAGVLTIALPVPVIVSNFNYFYHRETEGEEQAQYMHVGSCQHLSSSAEELRKARSNSTLSKSEYMVIEEGGMNHSAFPQTPFKTGNSTATCTTNNNPNSCVNIKKIFTDV