Reaction Details
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Target
Cyclic nucleotide-gated olfactory channel
Ligand
BDBM50526580
Substrate
n/a
Meas. Tech.
ChEMBL_1900214 (CHEMBL4402329)
EC50
6400±n/a nM
Citation
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More Info.:
Target
Name:
Cyclic nucleotide-gated olfactory channel
Synonyms:
CNG channel alpha-2 | CNG-2 | CNG2 | CNGA2_RAT | Cncg2 | Cnga2 | Cyclic nucleotide-gated cation channel 2 | Cyclic nucleotide-gated channel alpha-2 | Cyclic nucleotide-gated olfactory channel | Cyclic nucleotide-gated olfactory channel subunit OCNC1
Type:
PROTEIN
Mol. Mass.:
76176.63
Organism:
Rattus norvegicus
Description:
ChEMBL_119374
Residue:
664
Sequence:
MMTEKSNGVKSSPANNHNHHPPPSIKANGKDDHRAGSRPQSVAADDDTSPELQRLAEMDTPRRGRGGFQRIVRLVGVIRDWANKNFREEEPRPDSFLERFRGPELQTVTTHQGDDKGGKDGEGKGTKKKFELFVLDPAGDWYYRWLFVIAMPVLYNWCLLVARACFSDLQRNYFVVWLVLDYFSDTVYIADLIIRLRTGFLEQGLLVKDPKKLRDNYIHTLQFKLDVASIIPTDLIYFAVGIHSPEVRFNRLLHFARMFEFFDRTETRTSYPNIFRISNLVLYILVIIHWNACIYYVISKSIGFGVDTWVYPNITDPEYGYLAREYIYCLYWSTLTLTTIGETPPPVKDEEYLFVIFDFLIGVLIFATIVGNVGSMISNMNATRAEFQAKIDAVKHYMQFRKVSKDMEAKVIKWFDYLWTNKKTVDEREVLKNLPAKLRAEIAINVHLSTLKKVRIFQDCEAGLLVELVLKLRPQVFSPGDYICRKGDIGKEMYIIKEGKLAVVADDGVTQYALLSAGSCFGEISILNIKGSKMGNRRTANIRSLGYSDLFCLSKDDLMEAVTEYPDAKKVLEERGREILMKEGLLDENEVAASMEVDVQEKLEQLETNMDTLYTRFARLLAEYTGAQQKLKQRITVLETKMKQNHEDDYLSDGINTPEPTAAE