Reaction Details
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Target
Thiopurine S-methyltransferase
Ligand
BDBM50530712
Substrate
n/a
Meas. Tech.
ChEMBL_1913772 (CHEMBL4416355)
IC50
1000±n/a nM
Citation
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More Info.:
Target
Name:
Thiopurine S-methyltransferase
Synonyms:
TPMT | TPMT_HUMAN
Type:
PROTEIN
Mol. Mass.:
28178.47
Organism:
Homo sapiens (Human)
Description:
ChEMBL_1458987
Residue:
245
Sequence:
MDGTRTSLDIEEYSDTEVQKNQVLTLEEWQDKWVNGKTAFHQEQGHQLLKKHLDTFLKGKSGLRVFFPLCGKAVEMKWFADRGHSVVGVEISELGIQEFFTEQNLSYSEEPITEIPGTKVFKSSSGNISLYCCSIFDLPRTNIGKFDMIWDRGALVAINPGDRKCYADTMFSLLGKKFQYLLCVLSYDPTKHPGPPFYVPHAEIERLFGKICNIRCLEKVDAFEERHKSWGIDCLFEKLYLLTEK