Reaction Details
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Target
Serine palmitoyltransferase 1
Ligand
BDBM50535847
Substrate
n/a
Meas. Tech.
ChEMBL_1932328 (CHEMBL4477980)
IC50
64±n/a nM
Citation
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More Info.:
Target
Name:
Serine palmitoyltransferase 1
Synonyms:
LCB 1 | LCB1 | Long chain base biosynthesis protein 1 | SPT 1 | SPT1 | SPTC1_HUMAN | SPTLC1 | Serine-palmitoyl-CoA transferase 1
Type:
PROTEIN
Mol. Mass.:
52739.30
Organism:
Homo sapiens (Human)
Description:
ChEMBL_660503
Residue:
473
Sequence:
MATATEQWVLVEMVQALYEAPAYHLILEGILILWIIRLLFSKTYKLQERSDLTVKEKEELIEEWQPEPLVPPVPKDHPALNYNIVSGPPSHKTVVNGKECINFASFNFLGLLDNPRVKAAALASLKKYGVGTCGPRGFYGTFDVHLDLEDRLAKFMKTEEAIIYSYGFATIASAIPAYSKRGDIVFVDRAACFAIQKGLQASRSDIKLFKHNDMADLERLLKEQEIEDQKNPRKARVTRRFIVVEGLYMNTGTICPLPELVKLKYKYKARIFLEESLSFGVLGEHGRGVTEHYGINIDDIDLISANMENALASIGGFCCGRSFVIDHQRLSGQGYCFSASLPPLLAAAAIEALNIMEENPGIFAVLKEKCGQIHKALQGISGLKVVGESLSPAFHLQLEESTGSREQDVRLLQEIVDQCMNRSIALTQARYLEKEEKCLPPPSIRVVVTVEQTEEELERAASTIKEVAQAVLL