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Target
Casein kinase II subunit alpha 3
Ligand
BDBM50539770
Substrate
n/a
Meas. Tech.
ChEMBL_1979300 (CHEMBL4612435)
IC50
14±n/a nM
Citation
Rangasamy, L; Ortín, I; Zapico, JM; Coderch, C; Ramos, A; de Pascual-Teresa, B New Dual CK2/HDAC1 Inhibitors with Nanomolar Inhibitory Activity against Both Enzymes. ACS Med Chem Lett 11:713-719 (2020) [PubMed] Article
More Info.:
Target
Name:
Casein kinase II subunit alpha 3
Synonyms:
2.7.11.1 | CK II alpha 3 | CSK23_HUMAN | CSNK2A1P | CSNK2A3 | Casein kinase II alpha 1 polypeptide pseudogene | Casein kinase II subunit alpha 3
Type:
PROTEIN
Mol. Mass.:
45229.76
Organism:
Homo sapiens
Description:
ChEMBL_116899
Residue:
391
Sequence:
MSGPVPSRARVYTDVNTHRPREYWDYESHVVEWGNQDDYQLVRKLGRGKYSEVFEAINITNNEKVVVKILKPVKKKKIKREIKILENLRGGPNIITLADIVKDPVSRTPALVFEHVNNTDFKQLYQTLTDYDIRFYMYEILKALDYCHSMGIMHRDVKPHNVMIDHEHRKLRLIDWGLAEFYHPGQEYNVRVASRYFKGPELLVDYQMYDYSLDMWRLGCMLASMIFRKEPFFHGRDNYDQLVRIAKFLGTEDLYGYIDKYNIELDPRFNDILGRHSRKRWERFVHSENQHLVSPEALDFLDKLLRYDHQSRLTAREAMEHPYFYTVVKDQARMGSSSMPGGSTPVSSANVMSGISSVPTPSPLGPLAGSPVIAAANPLGMPVPAATGAQQ