Target
Serine/threonine-protein kinase ULK3
Ligand
BDBM50024294
Substrate
n/a
Meas. Tech.
ChEMBL_325004 (CHEMBL860640)
Kd
680±n/a nM
Citation
Target
Name:
Serine/threonine-protein kinase ULK3
Synonyms:
ULK3 kinase | ULK3_MOUSE | Ulk3
Type:
PROTEIN
Mol. Mass.:
53575.05
Organism:
Mus musculus
Description:
ChEMBL_325004
Residue:
472
Sequence:
MAGPSWGLPRLDGFILTERLGSGTYATVYKAYAKKDTREVVAIKCVAKKSLNKASVENLLTEIEILKGIRHPHIVQLKDFQWDNDNIYLIMEFCAGGDLSRFIHTRRILPEKVARVFMQQLASALQFLHERNISHLDLKPQNILLSSLEKPHLKLADFGFAQHMSPWDEKHVLRGSPLYMAPEMVCRRQYDARVDLWSVGVILYEALFGQPPFASRSFSELEEKIRSNRVIELPLRPQLSLDCRDLLQRLLERDPARRISFKDFFAHPWVDLEHMPSGESLAQARALVVEAVKKDQEGDAAAALSLYCKALDFFVPALHYEVDAQRKEAIKAKVGQYVSRAEELKAIVSSSNQALLRQGTTVQELLREMARDKPRLLAALEVASAALAKEEEAGKEQDALDLYQHSLGELLVLLAAEAPGRRRELLHTEVQNLMARAEYLKEQIKIRESHWEAESLDKEGLSESVRSSCTLQ
  
Inhibitor
Name:
BDBM50024294
Synonyms:
SP-600125
Type:
Small organic molecule
Emp. Form.:
C14H8N2O
Mol. Mass.:
220.2261
SMILES:
Oc1c2cccc3N=Nc(c23)c2ccccc12 |c:7|
Structure:
Search PDB for entries with ligand similarity: