Reaction Details
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Target
Potassium voltage-gated channel subfamily A member 2
Ligand
BDBM50182587
Substrate
n/a
Meas. Tech.
ChEMBL_334898 (CHEMBL861276)
EC50
2500±n/a nM
Citation
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More Info.:
Target
Name:
Potassium voltage-gated channel subfamily A member 2
Synonyms:
HBK5 | HUKIV | KCNA2 | KCNA2_HUMAN | NGK1 | Potassium voltage-gated channel subfamily A member 2 | Voltage-gated potassium channel | Voltage-gated potassium channel subunit Kv1.2
Type:
PROTEIN
Mol. Mass.:
56695.97
Organism:
Homo sapiens (Human)
Description:
ChEMBL_334898
Residue:
499
Sequence:
MTVATGDPADEAAALPGHPQDTYDPEADHECCERVVINISGLRFETQLKTLAQFPETLLGDPKKRMRYFDPLRNEYFFDRNRPSFDAILYYYQSGGRLRRPVNVPLDIFSEEIRFYELGEEAMEMFREDEGYIKEEERPLPENEFQRQVWLLFEYPESSGPARIIAIVSVMVILISIVSFCLETLPIFRDENEDMHGSGVTFHTYSNSTIGYQQSTSFTDPFFIVETLCIIWFSFEFLVRFFACPSKAGFFTNIMNIIDIVAIIPYFITLGTELAEKPEDAQQGQQAMSLAILRVIRLVRVFRIFKLSRHSKGLQILGQTLKASMRELGLLIFFLFIGVILFSSAVYFAEADERESQFPSIPDAFWWAVVSMTTVGYGDMVPTTIGGKIVGSLCAIAGVLTIALPVPVIVSNFNYFYHRETEGEEQAQYLQVTSCPKIPSSPDLKKSRSASTISKSDYMEIQEGVNNSNEDFREENLKTANCTLANTNYVNITKMLTDV