Reaction Details Report a problem with these data
Target
Adenosine receptor A3
Ligand
BDBM50608206
Substrate
n/a
Meas. Tech.
ChEMBL_2273263
Ki
>10000±n/a nM
Citation
Jacobson, KA; Salmaso, V; Suresh, RR; Tosh, DK Expanding the repertoire of methanocarba nucleosides from purinergic signaling to diverse targets. RSC Med Chem 12:1808-1825 (2021) [PubMed]
More Info.:
Target
Name:
Adenosine receptor A3
Synonyms:
A3AR | AA3R_MOUSE | Adenosine A3 receptor | Adora3 | Gpcr2
Type:
PROTEIN
Mol. Mass.:
36460.91
Organism:
Mus musculus
Description:
ChEMBL_1515686
Residue:
319
Sequence:
MEADNTTETDWLNITYITMEAAIGLCAVVGNMLVIWVVKLNPTLRTTTVYFIVSLALADIAVGVLVIPLAIAVSLQVKMHFYACLFMSCVLLIFTHASIMSLLAIAVHRYLRVKLTVRYRTVTTQRRIWLFLGLCWLVSFLVGLTPMFGWNRKATLASSQNSSTLLCHFRSVVSLDYMVFFSFITWILVPLVVMCIIYLDIFYIIRNKLSQNLTGFRETRAFYGREFKTAKSLFLVLFLFALCWLPLSIINFVSYFDVKIPDVAMCLGILLSHANSMMNPIVYACKIKKFKETYFLILRAVRLCQTSDSLDSNMEQTTE