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Target
Group 10 secretory phospholipase A2
Ligand
BDBM50274442
Substrate
n/a
Meas. Tech.
ChEMBL_537139 (CHEMBL989799)
IC50
>1600±n/a nM
Citation
 Oslund, RC; Cermak, N; Verlinde, CL; Gelb, MH Simplified YM-26734 inhibitors of secreted phospholipase A2 group IIA. Bioorg Med Chem Lett 18:5415-9 (2008) [PubMed]  Article
Target
Name:
Group 10 secretory phospholipase A2
Synonyms:
Group X secretory phospholipase A2 | PA2GX_MOUSE | Pla2g10
Type:
PROTEIN
Mol. Mass.:
17005.09
Organism:
Mus musculus
Description:
ChEMBL_537139
Residue:
151
Sequence:
MLLLLLLLLLGPGPGFSEATRRSHVYKRGLLELAGTLDCVGPRSPMAYMNYGCYCGLGGHGEPRDAIDWCCYHHDCCYSRAQDAGCSPKLDRYPWKCMDHHILCGPAENKCQELLCRCDEELAYCLAGTEYHLKYLFFPSILCEKDSPKCN
  
Inhibitor
Name:
BDBM50274442
Synonyms:
1-(3-Dodecanoyl-2-hydroxy-5-methyl-phenyl)-dodecan-1-one | CHEMBL484180
Type:
Small organic molecule
Emp. Form.:
C31H52O3
Mol. Mass.:
472.7428
SMILES:
CCCCCCCCCCCC(=O)c1cc(C)cc(C(=O)CCCCCCCCCCC)c1O
Structure:
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