Reaction Details
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Target
Vasoactive intestinal polypeptide receptor 1
Ligand
BDBM50366000
Substrate
n/a
Meas. Tech.
ChEMBL_807309 (CHEMBL1960402)
IC50
610±n/a nM
Citation
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More Info.:
Target
Name:
Vasoactive intestinal polypeptide receptor 1
Synonyms:
PACAP type II receptor | PACAP-R-2 | PACAP-R2 | Pituitary adenylate cyclase-activating polypeptide type II receptor | VIP-R-1 | VIPR1_RAT | Vipr1
Type:
PROTEIN
Mol. Mass.:
52068.73
Organism:
Rattus norvegicus
Description:
ChEMBL_807309
Residue:
459
Sequence:
MRPPSPPHVRWLCVLAGALACALRPAGSQAASPQHECEYLQLIEIQRQQCLEEAQLENETTGCSKMWDNLTCWPTTPRGQAVVLDCPLIFQLFAPIHGYNISRSCTEEGWSQLEPGPYHIACGLNDRASSLDEQQQTKFYNTVKTGYTIGYSLSLASLLVAMAILSLFRKLHCTRNYIHMHLFMSFILRATAVFIKDMALFNSGEIDHCSEASVGCKAAVVFFQYCVMANFFWLLVEGLYLYTLLAVSFFSERKYFWGYILIGWGVPSVFITIWTVVRIYFEDFGCWDTIINSSLWWIIKAPILLSILVNFVLFICIIRILVQKLRPPDIGKNDSSPYSRLAKSTLLLIPLFGIHYVMFAFFPDNFKAQVKMVFELVVGSFQGFVVAILYCFLNGEVQAELRRKWRRWHLQGVLGWSSKSQHPWGGSNGATCSTQVSMLTRVSPSARRSSSFQAEVSLV