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Target
Somatostatin receptor type 5
Ligand
BDBM50097781
Substrate
n/a
Meas. Tech.
ChEBML_200522
Ki
430±n/a nM
Citation
 Contour-Galéra, MO; Poitout, L; Moinet, C; Morgan, B; Gordon, T; Roubert, P; Thurieau, C Synthesis of substituted imidazopyrazines as ligands for the human somatostatin receptor subtype 5. Bioorg Med Chem Lett 11:741-5 (2001) [PubMed]
Target
Name:
Somatostatin receptor type 5
Synonyms:
SOMATOSTATIN SST5 | SS-5-R | SS5-R | SS5R | SSR5_HUMAN | SSTR5 | Somatostatin receptor type 5 (SSTR5)
Type:
Enzyme
Mol. Mass.:
39218.02
Organism:
Homo sapiens (Human)
Description:
P35346
Residue:
364
Sequence:
MEPLFPASTPSWNASSPGAASGGGDNRTLVGPAPSAGARAVLVPVLYLLVCAAGLGGNTLVIYVVLRFAKMKTVTNIYILNLAVADVLYMLGLPFLATQNAASFWPFGPVLCRLVMTLDGVNQFTSVFCLTVMSVDRYLAVVHPLSSARWRRPRVAKLASAAAWVLSLCMSLPLLVFADVQEGGTCNASWPEPVGLWGAVFIIYTAVLGFFAPLLVICLCYLLIVVKVRAAGVRVGCVRRRSERKVTRMVLVVVLVFAGCWLPFFTVNIVNLAVALPQEPASAGLYFFVVILSYANSCANPVLYGFLSDNFRQSFQKVLCLRKGSGAKDADATEPRPDRIRQQQEATPPAHRAAANGLMQTSKL
  
Inhibitor
Name:
BDBM50097781
Synonyms:
3-[6-(3-Nitro-phenyl)-2-phenyl-imidazo[1,2-a]pyrazin-8-yl]-propylamine | CHEMBL164964
Type:
Small organic molecule
Emp. Form.:
C21H19N5O2
Mol. Mass.:
373.4079
SMILES:
NCCCc1nc(cn2cc(nc12)-c1ccccc1)-c1cccc(c1)[N+]([O-])=O
Structure:
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