Target
Somatostatin receptor type 3
Ligand
BDBM50099170
Substrate
n/a
Meas. Tech.
ChEBML_225194
Ki
240±n/a nM
Citation
 Moinet, CContour-Galcéra, MOPoitout, LMorgan, BGordon, TRouber, PThurieau, C Novel non-peptide ligands for the somatostatin sst3 receptor. Bioorg Med Chem Lett 11:991-5 (2001) [PubMed]
Target
Name:
Somatostatin receptor type 3
Synonyms:
SOMATOSTATIN SST3 | SS-3-R | SS3-R | SS3R | SSR-28 | SSR3_HUMAN | SSTR3 | Somatostatin receptor type 3 (SSTR3)
Type:
Protein
Mol. Mass.:
45855.97
Organism:
Homo sapiens (Human)
Description:
P32745
Residue:
418
Sequence:
MDMLHPSSVSTTSEPENASSAWPPDATLGNVSAGPSPAGLAVSGVLIPLVYLVVCVVGLLGNSLVIYVVLRHTASPSVTNVYILNLALADELFMLGLPFLAAQNALSYWPFGSLMCRLVMAVDGINQFTSIFCLTVMSVDRYLAVVHPTRSARWRTAPVARTVSAAVWVASAVVVLPVVVFSGVPRGMSTCHMQWPEPAAAWRAGFIIYTAALGFFGPLLVICLCYLLIVVKVRSAGRRVWAPSCQRRRRSERRVTRMVVAVVALFVLCWMPFYVLNIVNVVCPLPEEPAFFGLYFLVVALPYANSCANPILYGFLSYRFKQGFRRVLLRPSRRVRSQEPTVGPPEKTEEEDEEEEDGEESREGGKGKEMNGRVSQITQPGTSGQERPPSRVASKEQQLLPQEASTGEKSSTMRISYL
  
Inhibitor
Name:
BDBM50099170
Synonyms:
CHEMBL368993 | N-[(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-2-(3-trifluoromethyl-phenyl)-acetamide
Type:
Small organic molecule
Emp. Form.:
C28H23F3N4O
Mol. Mass.:
488.5036
SMILES:
FC(F)(F)c1cccc(CC(=O)N[C@H](Cc2c[nH]c3ccccc23)c2nc(c[nH]2)-c2ccccc2)c1
Structure:
Search PDB for entries with ligand similarity: