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Target
Somatostatin receptor type 1
Ligand
BDBM50099181
Substrate
n/a
Meas. Tech.
ChEBML_225192
Ki
1400±n/a nM
Citation
 Moinet, C; Contour-Galcéra, MO; Poitout, L; Morgan, B; Gordon, T; Rouber, P; Thurieau, C Novel non-peptide ligands for the somatostatin sst3 receptor. Bioorg Med Chem Lett 11:991-5 (2001) [PubMed]
Target
Name:
Somatostatin receptor type 1
Synonyms:
SOMATOSTATIN SST1 | SRIF-2 | SS-1-R | SS1-R | SS1R | SSR1_HUMAN | SSTR1 | Somatostatin receptor type 1 (SSTR1)
Type:
Enzyme
Mol. Mass.:
42692.81
Organism:
Homo sapiens (Human)
Description:
P30872
Residue:
391
Sequence:
MFPNGTASSPSSSPSPSPGSCGEGGGSRGPGAGAADGMEEPGRNASQNGTLSEGQGSAILISFIYSVVCLVGLCGNSMVIYVILRYAKMKTATNIYILNLAIADELLMLSVPFLVTSTLLRHWPFGALLCRLVLSVDAVNMFTSIYCLTVLSVDRYVAVVHPIKAARYRRPTVAKVVNLGVWVLSLLVILPIVVFSRTAANSDGTVACNMLMPEPAQRWLVGFVLYTFLMGFLLPVGAICLCYVLIIAKMRMVALKAGWQQRKRSERKITLMVMMVVMVFVICWMPFYVVQLVNVFAEQDDATVSQLSVILGYANSCANPILYGFLSDNFKRSFQRILCLSWMDNAAEEPVDYYATALKSRAYSVEDFQPENLESGGVFRNGTCTSRITTL
  
Inhibitor
Name:
BDBM50099181
Synonyms:
CHEMBL177337 | [(R)-2-(1H-Indol-3-yl)-1-(4-phenyl-1H-imidazol-2-yl)-ethyl]-carbamic acid benzyl ester
Type:
Small organic molecule
Emp. Form.:
C27H24N4O2
Mol. Mass.:
436.5051
SMILES:
O=C(N[C@H](Cc1c[nH]c2ccccc12)c1nc(c[nH]1)-c1ccccc1)OCc1ccccc1
Structure:
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