Reaction Details
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Target
Pyruvate kinase PKLR
Ligand
BDBM50367050
Substrate
n/a
Meas. Tech.
ChEMBL_160246 (CHEMBL767860)
Ki
8000000±n/a nM
Citation
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More Info.:
Target
Name:
Pyruvate kinase PKLR
Synonyms:
KPYR_RAT | Pklr | Pyruvate kinase isozymes R/L
Type:
PROTEIN
Mol. Mass.:
62202.26
Organism:
Rattus norvegicus
Description:
ChEMBL_1359662
Residue:
574
Sequence:
MSVQENTLPQQLWPWIFRSQKDLAKSALSGAPGGPAGYLRRASVAQLTQELGTAFFQQQQLPAAMADTFLEHLCLLDIDSQPVAARSTSIIATIGPASRSVDRLKEMIKAGMNIARLNFSHGSHEYHAESIANIREATESFATSPLSYRPVAIALDTKGPEIRTGVLQGGPESEVEIVKGSQVLVTVDPKFQTRGDAKTVWVDYHNITRVVAVGGRIYIDDGLISLVVQKIGPEGLVTEVEHGGILGSRKGVNLPNTEVDLPGLSEQDLLDLRFGVQHNVDIIFASFVRKASDVLAVRDALGPEGQNIKIISKIENHEGVKKFDEILEVSDGIMVARGDLGIEIPAEKVFLAQKMMIGRCNLAGKPVVCATQMLESMITKARPTRAETSDVANAVLDGADCIMLSGETAKGSFPVEAVMMQHAIAREAEAAVYHRQLFEELRRAAPLSRDPTEVTAIGAVEASFKCCAAAIIVLTKTGRSAQLLSQYRPRAAVIAVTRSAQAARQVHLSRGVFPLLYREPPEAIWADDVDRRVQFGIESGKLRGFLRVGDLVIVVTGWRPGSGYTNIMRVLSVS