Reaction Details
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Target
Pyruvate kinase PKM
Ligand
BDBM50367050
Substrate
n/a
Meas. Tech.
ChEMBL_160380 (CHEMBL765726)
Ki
4500000±n/a nM
Citation
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More Info.:
Target
Name:
Pyruvate kinase PKM
Synonyms:
KPYM_RAT | Pkm | Pkm2 | Pykm | Pyruvate kinase isozymes M1/M2
Type:
PROTEIN
Mol. Mass.:
57820.70
Organism:
Rattus norvegicus
Description:
ChEMBL_160255
Residue:
531
Sequence:
MPKPDSEAGTAFIQTQQLHAAMADTFLEHMCRLDIDSAPITARNTGIICTIGPASRSVEMLKEMIKSGMNVARLNFSHGTHEYHAETIKNVRAATESFASDPILYRPVAVALDTKGPEIRTGLIKGSGTAEVELKKGATLKITLDNAYMEKCDENILWLDYKNICKVVEVGSKIYVDDGLISLQVKEKGADYLVTEVENGGSLGSKKGVNLPGAAVDLPAVSEKDIQDLKFGVEQDVDMVFASFIRKAADVHEVRKVLGEKGKNIKIISKIENHEGVRRFDEILEASDGIMVARGDLGIEIPAEKVFLAQKMMIGRCNRAGKPVICATQMLESMIKKPRPTRAEGSDVANAVLDGADCIMLSGETAKGDYPLEAVRMQHLIAREAEAAVFHRLLFEELARASSQSTDPLEAMAMGSVEASYKCLAAALIVLTESGRSAHQVARYRPRAPIIAVTRNPQTARQAHLYRGIFPVLCKDAVLDAWAEDVDLRVNLAMNVGKARGFFKKGDVVIVLTGWRPGSGFTNTMRVVPVP