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Target
Mu-type opioid receptor
Ligand
BDBM50422811
Substrate
n/a
Meas. Tech.
ChEMBL_334063 (CHEMBL861853)
IC50
200±n/a nM
Citation
 Middleton, DS; Maw, GN; Challenger, C; Jessiman, A; Johnson, PS; Million, WA; Nichols, CL; Price, JA; Trevethick, M Highly potent and selective zwitterionic agonists of the delta-opioid receptor. Part 1. Bioorg Med Chem Lett 16:905-10 (2006) [PubMed]  Article
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50422811
Synonyms:
CHEMBL204716
Type:
Small organic molecule
Emp. Form.:
C31H35N3O4
Mol. Mass.:
513.6273
SMILES:
C[C@@H]1CN([C@@H](c2cccc(O)c2)c2ccc3CCN(Cc3c2)C(=O)C(O)=O)[C@@H](C)CN1Cc1ccccc1
Structure:
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