Reaction Details Report a problem with these data
Target
Kinesin-like protein KIFC1
Ligand
BDBM50037899
Substrate
n/a
Meas. Tech.
ChEMBL_1438848 (CHEMBL3390316)
IC50
37000±n/a nM
Citation
Yang, B; Lamb, ML; Zhang, T; Hennessy, EJ; Grewal, G; Sha, L; Zambrowski, M; Block, MH; Dowling, JE; Su, N; Wu, J; Deegan, T; Mikule, K; Wang, W; Kaspera, R; Chuaqui, C; Chen, H Discovery of potent KIFC1 inhibitors using a method of integrated high-throughput synthesis and screening. J Med Chem 57:9958-70 (2014) [PubMed] Article
More Info.:
Target
Name:
Kinesin-like protein KIFC1
Synonyms:
HSET | HSET | KIFC1 | KIFC1_HUMAN | KNSL2 | Kinesin-like protein 2 | Kinesin-like protein KIFC1 | Kinesin-related protein HSET
Type:
PROTEIN
Mol. Mass.:
73763.89
Organism:
Homo sapiens (Human)
Description:
ChEMBL_109524
Residue:
673
Sequence:
MDPQRSPLLEVKGNIELKRPLIKAPSQLPLSGSRLKRRPDQMEDGLEPEKKRTRGLGATTKITTSHPRVPSLTTVPQTQGQTTAQKVSKKTGPRCSTAIATGLKNQKPVPAVPVQKSGTSGVPPMAGGKKPSKRPAWDLKGQLCDLNAELKRCRERTQTLDQENQQLQDQLRDAQQQVKALGTERTTLEGHLAKVQAQAEQGQQELKNLRACVLELEERLSTQEGLVQELQKKQVELQEERRGLMSQLEEKERRLQTSEAALSSSQAEVASLRQETVAQAALLTEREERLHGLEMERRRLHNQLQELKGNIRVFCRVRPVLPGEPTPPPGLLLFPSGPGGPSDPPTRLSLSRSDERRGTLSGAPAPPTRHDFSFDRVFPPGSGQDEVFEEIAMLVQSALDGYPVCIFAYGQTGSGKTFTMEGGPGGDPQLEGLIPRALRHLFSVAQELSGQGWTYSFVASYVEIYNETVRDLLATGTRKGQGGECEIRRAGPGSEELTVTNARYVPVSCEKEVDALLHLARQNRAVARTAQNERSSRSHSVFQLQISGEHSSRGLQCGAPLSLVDLAGSERLDPGLALGPGERERLRETQAINSSLSTLGLVIMALSNKESHVPYRNSKLTYLLQNSLGGSAKMLMFVNISPLEENVSESLNSLRFASKVNQCVIGTAQANRK