Reaction Details
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Target
UDP-glucuronosyltransferase 1A8
Ligand
BDBM50088502
Substrate
n/a
Meas. Tech.
ChEMBL_1489265 (CHEMBL3533108)
Ki
22600±n/a nM
Citation
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More Info.:
Target
Name:
UDP-glucuronosyltransferase 1A8
Synonyms:
GNT1 | GNT1 | UD18_HUMAN | UDP-glucuronosyltransferase 1-8 | UDP-glucuronosyltransferase 1-H | UDP-glucuronosyltransferase 1A8 | UDPGT 1-8 | UGT-1H | UGT1 | UGT1*8 | UGT1-08 | UGT1.8 | UGT1A8 | UGT1H
Type:
PROTEIN
Mol. Mass.:
59751.98
Organism:
Homo sapiens (Human)
Description:
ChEMBL_104086
Residue:
530
Sequence:
MARTGWTSPIPLCVSLLLTCGFAEAGKLLVVPMDGSHWFTMQSVVEKLILRGHEVVVVMPEVSWQLGKSLNCTVKTYSTSYTLEDLDREFMDFADAQWKAQVRSLFSLFLSSSNGFFNLFFSHCRSLFNDRKLVEYLKESSFDAVFLDPFDACGLIVAKYFSLPSVVFARGIACHYLEEGAQCPAPLSYVPRILLGFSDAMTFKERVRNHIMHLEEHLFCQYFSKNALEIASEILQTPVTAYDLYSHTSIWLLRTDFVLDYPKPVMPNMIFIGGINCHQGKPLPMEFEAYINASGEHGIVVFSLGSMVSEIPEKKAMAIADALGKIPQTVLWRYTGTRPSNLANNTILVKWLPQNDLLGHPMTRAFITHAGSHGVYESICNGVPMVMMPLFGDQMDNAKRMETKGAGVTLNVLEMTSEDLENALKAVINDKSYKENIMRLSSLHKDRPVEPLDLAVFWVEFVMRHKGAPHLRPAAHDLTWYQYHSLDVIGFLLAVVLTVAFITFKCCAYGYRKCLGKKGRVKKAHKSKTH