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Target
Putative P2Y purinoceptor 10
Ligand
BDBM50096349
Substrate
n/a
Meas. Tech.
ChEMBL_1581711 (CHEMBL3816044)
EC50
25±n/a nM
Citation
 Jung, S; Inoue, A; Nakamura, S; Kishi, T; Uwamizu, A; Sayama, M; Ikubo, M; Otani, Y; Kano, K; Makide, K; Aoki, J; Ohwada, T Conformational Constraint of the Glycerol Moiety of Lysophosphatidylserine Affords Compounds with Receptor Subtype Selectivity. J Med Chem 59:3750-76 (2016) [PubMed]  Article
Target
Name:
Putative P2Y purinoceptor 10
Synonyms:
P2Y10 | P2Y10_MOUSE | P2ry10 | Putative P2Y purinoceptor 10
Type:
PROTEIN
Mol. Mass.:
37264.07
Organism:
Mus musculus
Description:
ChEMBL_109764
Residue:
328
Sequence:
MGSNSTSSAESNCNATYLPFQYSLYATTYIFIFIPGLLANSAALWVLCRFISKKNKAIIFMINLSVADLAHILSLPLRIYYYINRHWPFQRALCLLCFYLKYLNMYASIFFLTCISLQRCLFLLKPFRARNWKRRYDVGISAVIWIVVGTACLPFPILRNAGLANSTDSCFADLGYKQMDAVVLVTMVVIAELAGFVIPVITIACCTWKTTVSLKHPPIAFQGISERKKALRMVFMCAAVFVICFTPYHINFIFYTMVKESIITSCPTVKSTLYFHPFSLCLASLCCLLDPILYYFMASEFRDQLSRHGSSVTRSRLMSRESGSSMVN
  
Inhibitor
Name:
BDBM50096349
Synonyms:
CHEBI:52649 | CHEMBL1742484
Type:
Small organic molecule
Emp. Form.:
C24H46NO9P
Mol. Mass.:
523.5971
SMILES:
CCCCCCCC\C=C/CCCCCCCC(=O)OC[C@@H](O)COP(O)(=O)OC[C@H](N)C(O)=O |r|
Structure:
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