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Target
Beta-lactamase BRO-1
Ligand
BDBM50212640
Substrate
n/a
Meas. Tech.
ChEMBL_40225 (CHEMBL653998)
IC50
2.89±n/a nM
Citation
TBA Bioorg Med Chem Lett 3:2247-2252 (1993)
More Info.:
Target
Name:
Beta-lactamase BRO-1
Synonyms:
BLA1_MORCA | Beta-lactamase BRO-1 | Penicillinase | bla
Type:
PROTEIN
Mol. Mass.:
35383.81
Organism:
Moraxella catarrhalis
Description:
ChEMBL_104100
Residue:
313
Sequence:
MQRRHFLQKTLLALPIIFSGNLLTGCKTNLSDDYLPDDKITNNPNLLQNKLKEILPIWENKFNAKIGMTIIADNGELSSHRGNEYFPVNSTIKAFIASHILLLVDKEKLDLNEKIIIKESDLIEYSPVCKKYFDENKPISISELCEATITLSDNGSANILLDKIGGLTAFNQFLKEIGADMVLANNEPLLNRSHYGETSDTAKPIPYTKSLKALIVGNILSNQSKEQLITWLINDKVADNLLRKYLPKNWRIGDKTGTGSESKNIIAVIWNENNKPYFISLFITQPHDGKSLDFKNQKDEIMAQIGKEIYPFL