Reaction Details 
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Report a problem with these dataTarget
Melatonin receptor
Ligand
BDBM85058
Substrate
n/a
Ki
1.6±n/a nM
Comments
PDSP_120
Citation
Dubocovich, ML; Masana, MI; Iacob, S; Sauri, DM Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor. Naunyn Schmiedebergs Arch Pharmacol 355:365-75 (1997) [PubMed] ArticleMore Info.:
Target
Name:
Melatonin receptor
Synonyms:
Melatonin | Melatonin receptor
Type:
Enzyme Catalytic Domain
Mol. Mass.:
13287.02
Organism:
RABBIT
Description:
Q9BE38
Residue:
114
Sequence:
MIWMLTLVAVMPNLHTGTLQYDPRVYSCTFSQSVSSAYTIAVVVFHFIIPMLMSSCCYLRIWILVLQVRRRVKPDNKPKLKPQDFRNFITMFVVFVLFAICWAPLNFIVLLGRS
Inhibitor
Name:
BDBM85058
Synonyms:
4-P-ADOT | 4-phenyl-2-acetamidotetraline
Type:
Small organic molecule
Emp. Form.:
C18H19NO
Mol. Mass.:
265.3496
SMILES:
CC(=O)NC1CC(c2ccccc2)c2ccccc2C1
Structure:
