Target
Neuropeptide Y receptor type 2
Ligand
BDBM84998
Substrate
n/a
Ki
3.22±n/a nM
Comments
PDSP_1372
Citation
 Sharma, PHolmberg, SKEriksson, HBeck-Sickinger, AGGrundemar, LLarhammar, D Cloning and functional expression of the guinea pig neuropeptide Y Y2 receptor. Regul Pept 0:23-8 (1998) [PubMed]  Article
Target
Name:
Neuropeptide Y receptor type 2
Synonyms:
NPY-Y2 | NPY2R | NPY2R_CAVPO | Neuropeptide Y receptor type 2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42344.53
Organism:
GUINEA PIG
Description:
NPY-Y2 NPY2R GUINEA PIG::Q9Z2D5
Residue:
381
Sequence:
MGPIGTEADENQTVEEIKVEPYGPGHTTPRGELAPDPEPELIDSTKLTEVRVVLILAYCSIILLGVVGNSLVIHVVIKFKSMRTVTNFFIANLAVADLLVNTLCLPFTLTYTLMGEWKMGPVLCHLVPYAQGLAVQVSTVTLTVIALDRHRCIVYHLDSKISKQNSFLIIGLAWGISALLASPLAIFREYSLIEIIPDFEIVACTEKWPGEEKSIYGTVYSLSSLLILYVLPLGIISVSYVRIWSKLKNHVSPGAANDHYHQRRQKTTKMLVFVVVVFAVSWLPLHAFQLAVDIDSQVLDLKEYKLIFTVFHIIAMCSTFANPLLYGWMNSNYRKAFLSAFRCQQRLDAIQSEVCVTGKAKTNVEVEKNHGAADSAEATNV
  
Inhibitor
Name:
BDBM84998
Synonyms:
NPY 3-36, porcine
Type:
Small organic molecule
Emp. Form.:
C195H295N53O57
Mol. Mass.:
4293.7497
SMILES:
n/a
Structure:
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