Reaction Details  Report a problem with these data
Target
Somatostatin receptor type 2
Ligand
BDBM85520
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_3370
Citation
 Reubi, JC; Schaer, JC; Wenger, S; Hoeger, C; Erchegyi, J; Waser, B; Rivier, J SST3-selective potent peptidic somatostatin receptor antagonists. Proc Natl Acad Sci U S A 97:13973-8 (2000) [PubMed]  Article
Target
Name:
Somatostatin receptor type 2
Synonyms:
SOMATOSTATIN SST2 | SRIF-1 | SS-2-R | SS2-R | SS2R | SSR2_HUMAN | SSTR2 | Somatostatin receptor type 2 (SSTR2)
Type:
Enzyme
Mol. Mass.:
41344.94
Organism:
Homo sapiens (Human)
Description:
P30874
Residue:
369
Sequence:
MDMADEPLNGSHTWLSIPFDLNGSVVSTNTSNQTEPYYDLTSNAVLTFIYFVVCIIGLCGNTLVIYVILRYAKMKTITNIYILNLAIADELFMLGLPFLAMQVALVHWPFGKAICRVVMTVDGINQFTSIFCLTVMSIDRYLAVVHPIKSAKWRRPRTAKMITMAVWGVSLLVILPIMIYAGLRSNQWGRSSCTINWPGESGAWYTGFIIYTFILGFLVPLTIICLCYLFIIIKVKSSGIRVGSSKRKKSEKKVTRMVSIVVAVFIFCWLPFYIFNVSSVSMAISPTPALKGMFDFVVVLTYANSCANPILYAFLSDNFKKSFQNVLCLVKVSGTDDGERSDSKQDKSRLNETTETQRTLLNGDLQTSI
  
Inhibitor
Name:
BDBM85520
Synonyms:
CAS_5311373 | L-796,778 | NSC_5311373
Type:
Small organic molecule
Emp. Form.:
C29H40N6O7
Mol. Mass.:
584.6639
SMILES:
CCCCC(NC(=O)NC(Cc1ccccc1)C(=O)Nc1ccc(cc1)[N+]([O-])=O)C(=O)NC(CCCCN)C(=O)OC
Structure:
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