Reaction Details  Report a problem with these data
Target
Cannabinoid receptor 1
Ligand
BDBM85795
Substrate
n/a
Ki
53±n/a nM
Comments
PDSP_1398
Citation
 Breivogel, CS; Griffin, G; Di Marzo, V; Martin, BR Evidence for a new G protein-coupled cannabinoid receptor in mouse brain. Mol Pharmacol 60:155-63 (2001) [PubMed]
Target
Name:
Cannabinoid receptor 1
Synonyms:
Brain-type cannabinoid receptor | CANNABINOID CB1 | CB-R | CB1 | CNR1_RAT | Cannabinoid CB1 receptor | Cannabinoid receptor | Cannabinoid receptor 1 (CB1) | Cnr1 | Skr6
Type:
G Protein-Coupled Receptor (GPCR)
Mol. Mass.:
52856.55
Organism:
Rattus norvegicus (rat)
Description:
P20272
Residue:
473
Sequence:
MKSILDGLADTTFRTITTDLLYVGSNDIQYEDIKGDMASKLGYFPQKFPLTSFRGSPFQEKMTAGDNSPLVPAGDTTNITEFYNKSLSSFKENEENIQCGENFMDMECFMILNPSQQLAIAVLSLTLGTFTVLENLLVLCVILHSRSLRCRPSYHFIGSLAVADLLGSVIFVYSFVDFHVFHRKDSPNVFLFKLGGVTASFTASVGSLFLTAIDRYISIHRPLAYKRIVTRPKAVVAFCLMWTIAIVIAVLPLLGWNCKKLQSVCSDIFPLIDETYLMFWIGVTSVLLLFIVYAYMYILWKAHSHAVRMIQRGTQKSIIIHTSEDGKVQVTRPDQARMDIRLAKTLVLILVVLIICWGPLLAIMVYDVFGKMNKLIKTVFAFCSMLCLLNSTVNPIIYALRSKDLRHAFRSMFPSCEGTAQPLDNSMGDSDCLHKHANNTASMHRAAESCIKSTVKIAKVTMSVSTDTSAEAL
  
Inhibitor
Name:
BDBM85795
Synonyms:
(5Z,8Z,11Z,14Z)-2-Methyl-N-(2-hydroxyethyl)-5,8,11,14-icosatetrenamide | O-680
Type:
Small organic molecule
Emp. Form.:
C23H39NO2
Mol. Mass.:
361.5613
SMILES:
CCCCC\C=C\C\C=C\C\C=C\C\C=C\CCC(C)C(=O)NCCO
Structure:
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