Reaction Details 
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Report a problem with these dataTarget
Norepinephrine transporter
Ligand
BDBM50021952
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_283
Citation
Davids, E; Zhang, K; Kula, NS; Tarazi, FI; Baldessarini, RJ Effects of norepinephrine and serotonin transporter inhibitors on hyperactivity induced by neonatal 6-hydroxydopamine lesioning in rats. J Pharmacol Exp Ther 301:1097-102 (2002) [PubMed] ArticleMore Info.:
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
Inhibitor
Name:
BDBM50021952
Synonyms:
7-Benzyl-1-ethyl-4-oxo-1,4-dihydro-[1,8]naphthyridine-3-carboxylic acid | Amfonelic acid | CHEMBL35337
Type:
Small organic molecule
Emp. Form.:
C18H16N2O3
Mol. Mass.:
308.3312
SMILES:
CCn1cc(C(O)=O)c(=O)c2ccc(Cc3ccccc3)nc12
Structure:
