Target
Norepinephrine transporter
Ligand
BDBM50062915
Substrate
n/a
Ki
126±n/a nM
Comments
PDSP_2246
Citation
 Davids, EZhang, KKula, NSTarazi, FIBaldessarini, RJ Effects of norepinephrine and serotonin transporter inhibitors on hyperactivity induced by neonatal 6-hydroxydopamine lesioning in rats. J Pharmacol Exp Ther 301:1097-102 (2002) [PubMed]  Article
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
  
Inhibitor
Name:
BDBM50062915
Synonyms:
CHEMBL827 | METHYLPHENIDATE | methyl (2R)-phenyl[(2R)-piperidin-2-yl]acetate | methyl (R)-phenyl[(R)-piperidin-2-yl]acetate
Type:
Small organic molecule
Emp. Form.:
C14H19NO2
Mol. Mass.:
233.3062
SMILES:
COC(=O)[C@@H]([C@H]1CCCCN1)c1ccccc1
Structure:
Search PDB for entries with ligand similarity: