Reaction Details
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Target
Corticotropin-releasing factor receptor 1
Ligand
BDBM86058
Substrate
n/a
Ki
1000±n/a nM
Comments
PDSP_3044
Citation
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More Info.:
Target
Name:
Corticotropin-releasing factor receptor 1
Synonyms:
CRF1 | CRFR1_MACMU | CRHR1 | Corticotropin releasing hormone receptor type 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
47810.67
Organism:
Monkey
Description:
Q76LL8
Residue:
415
Sequence:
MARHPQLRLVKALLLLGLNPVSASLQDQHCESLSLASNISGLQCNASVDLIGTCWPRSPAGQLVVRPCPAFFYGVRYNTTNNGYRECLANGSWAARVNYSECQEILNEEKKSKVHYHVAVIINYLGHCISLVALLVAFVLFLRLRSIRCLRNIIHWNLISAFILRNATWFVVQLTMSPEVHQSNVGWCRLVTAAYNYFHVTNFFWMFGEGCYLHTAIVLTYSTDRLRKWMFICIGWGVPFPIIVAWAIGKLYYDNEKCWFGKRPGVYTDYIYQGPMILVLLINFIFLFNIVRILMTKLRASTTSETIQYRKAVKATLVLLPLLGITYMLFFVNPGEDEVSRVVFIYFNSFLESFQGFFVSVFYCFLNSEVRSAIRKRWHRWQDKHSIRARVARAMSIPTSPTRVSFHSIKQSTAV