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Target
Calcium-activated potassium channel subunit beta
Ligand
BDBM86247
Substrate
n/a
Ki
16±n/a nM
Comments
PDSP_3711
Citation
 Davis-Taber, R; Molinari, EJ; Altenbach, RJ; Whiteaker, KL; Shieh, CC; Rotert, G; Buckner, SA; Malysz, J; Milicic, I; McDermott, JS; Gintant, GA; Coghlan, MJ; Carroll, WA; Scott, VE; Gopalakrishnan, M [125I]A-312110, a novel high-affinity 1,4-dihydropyridine ATP-sensitive K+ channel opener: characterization and pharmacology of binding. Mol Pharmacol 64:143-53 (2003) [PubMed]  Article
Target
Name:
Calcium-activated potassium channel subunit beta
Synonyms:
Potassium channel (ATP modulatory)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
22836.62
Organism:
GUINEA PIG
Description:
C0KY85
Residue:
199
Sequence:
GSHAKPFMLSTQREESNCTIIHTHIMDDWMDCAFTCGVDCQGQGKYPCLQVFVNLTHSGQKALLHYNEEAVQINSKCFYTPKCRRDGNDLLNSALNIKEFFDHKNRTPFSCFYSPDNQSEDVILIKKYDQMVIFHCLFWPSMTMLGGALIVGMVRLTQYLFLLCEKYSTALRDEVSGKVPYVARNQFKLWSVGRSKGRA
  
Inhibitor
Name:
BDBM86247
Synonyms:
BAY X 9228 | CAS_3038059 | NSC_3038059
Type:
Small organic molecule
Emp. Form.:
C16H25N3O3
Mol. Mass.:
307.388
SMILES:
CCOc1ccccc1N=C(C[N+]([O-])=O)NC(C)C(C)(C)C |w:9.9|
Structure:
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