Reaction Details
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Target
Genome polyprotein [1027-1206,R1052K]
Ligand
BDBM92407
Substrate
n/a
Meas. Tech.
Binding Assay
pH
8±0
Ki
0.53±0.05 nM
KOFF
4.4E-4 s-1
KON
8.5E5 M-1s-1
Citation
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More Info.:
Target
Name:
Genome polyprotein [1027-1206,R1052K]
Synonyms:
HCV NS3 Proteinase | NS3-NS4A Protein | POLG_HCVCO
Type:
Enzyme Subunit
Mol. Mass.:
18947.03
Organism:
Hepatitis C virus
Description:
HCV (BK strain) NS3 protein region from amino acid 1 to 180, harboring a C-terminal poly Lys solubilization motif (ASKKKK).
Residue:
180
Sequence:
APITAYSQQTRGLLGCIITSLTGRDKNQVEGEVQVVSTATQSFLATCVNGVCWTVYHGAGSKTLAGPKGPITQMYTNVDQDLVGWQAPPGARSLTPCTCGSSDLYLVTRHADVIPVRRRGDSRGSLLSPRPVSYLKGSSGGPLLCPSGHAVGIFRAAVCTRGVAKAVDFVPVESMETTMR