Reaction Details
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Target
Phosphatidylcholine-sterol acyltransferase
Ligand
BDBM92616
Substrate
n/a
Meas. Tech.
Enzyme Assay
pH
7.5±0
Temperature
277.15±0 K
IC50
60±0.0 nM
Citation
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More Info.:
Target
Name:
Phosphatidylcholine-sterol acyltransferase
Synonyms:
LCAT | LCAT_HUMAN | Lecithin-cholesterol acyltransferase (LCAT) | Phospholipid-cholesterol acyltransferase
Type:
Protein
Mol. Mass.:
49573.79
Organism:
Homo sapiens (Human)
Description:
P04180
Residue:
440
Sequence:
MGPPGSPWQWVTLLLGLLLPPAAPFWLLNVLFPPHTTPKAELSNHTRPVILVPGCLGNQLEAKLDKPDVVNWMCYRKTEDFFTIWLDLNMFLPLGVDCWIDNTRVVYNRSSGLVSNAPGVQIRVPGFGKTYSVEYLDSSKLAGYLHTLVQNLVNNGYVRDETVRAAPYDWRLEPGQQEEYYRKLAGLVEEMHAAYGKPVFLIGHSLGCLHLLYFLLRQPQAWKDRFIDGFISLGAPWGGSIKPMLVLASGDNQGIPIMSSIKLKEEQRITTTSPWMFPSRMAWPEDHVFISTPSFNYTGRDFQRFFADLHFEEGWYMWLQSRDLLAGLPAPGVEVYCLYGVGLPTPRTYIYDHGFPYTDPVGVLYEDGDDTVATRSTELCGLWQGRQPQPVHLLPLHGIQHLNMVFSNLTLEHINAILLGAYRQGPPASPTASPEPPPPE