Reaction Details Report a problem with these data
Target
Diacylglycerol O-acyltransferase 1 [89-488]
Ligand
BDBM120755
Substrate
n/a
Meas. Tech.
Inhibition Assay
pH
7.5±n/a
Temperature
277.15±n/a K
IC50
8.5±n/a nM
Comments
extracted
Citation
Forster, CJ; Kwak, Y; Nakajima, K; Wang, B Organic compounds US Patent US8703761 Publication Date 4/22/2014
More Info.:
Target
Name:
Diacylglycerol O-acyltransferase 1 [89-488]
Synonyms:
AGRP1 | DGAT | DGAT1 | DGAT1_HUMAN | acyl coA-diacylglycerol acyl transferase 1 (DGAT1)
Type:
Protein
Mol. Mass.:
46366.89
Organism:
Homo sapiens (Human)
Description:
O75907[89-488]
Residue:
400
Sequence:
LNWCVVMLILSNARLFLENLIKYGILVDPIQVVSLFLKDPYSWPAPCLVIAANVFAVAAFQVEKRLAVGALTEQAGLLLHVANLATILCFPAAVVLLVESITPVGSLLALMAHTILFLKLFSYRDVNSWCRRARAKAASAGKKASSAAAPHTVSYPDNLTYRDLYYFLFAPTLCYELNFPRSPRIRKRFLLRRILEMLFFTQLQVGLIQQWMVPTIQNSMKPFKDMDYSRIIERLLKLAVPNHLIWLIFFYWLFHSCLNAVAELMQFGDREFYRDWWNSESVTYFWQNWNIPVHKWCIRHFYKPMLRRGSSKWMARTGVFLASAFFHEYLVSVPLRMFRLWAFTGMMAQIPLAWFVGRFFQGNYGNAAVWLSLIIGQPIAVLMYVHDYYVLNYEAPAAEA