Reaction Details
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Target
Isocitrate dehydrogenase [NADP], mitochondrial [R172S]
Ligand
BDBM195602
Substrate
n/a
Meas. Tech.
RapidFire-MS/MS and NADPH Assays
Temperature
298.15±n/a K
IC50
>100000±0.0 nM
Comments
extracted
Citation
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More Info.:
Target
Name:
Isocitrate dehydrogenase [NADP], mitochondrial [R172S]
Synonyms:
IDH2 | IDHP_HUMAN | Isocitrate dehydrogenase 2 mutant (R172S)
Type:
Protein
Mol. Mass.:
50853.19
Organism:
Homo sapiens (Human)
Description:
R172S mutant
Residue:
452
Sequence:
MAGYLRVVRSLCRASGSRPAWAPAALTAPTSQEQPRRHYADKRIKVAKPVVEMDGDEMTRIIWQFIKEKLILPHVDIQLKYFDLGLPNRDQTDDQVTIDSALATQKYSVAVKCATITPDEARVEEFKLKKMWKSPNGTIRNILGGTVFREPIICKNIPRLVPGWTKPITIGSHAHGDQYKATDFVADRAGTFKMVFTPKDGSGVKEWEVYNFPAGGVGMGMYNTDESISGFAHSCFQYAIQKKWPLYMSTKNTILKAYDGRFKDIFQEIFDKHYKTDFDKNKIWYEHRLIDDMVAQVLKSSGGFVWACKNYDGDVQSDILAQGFGSLGLMTSVLVCPDGKTIEAEAAHGTVTRHYREHQKGRPTSTNPIASIFAWTRGLEHRGKLDGNQDLIRFAQMLEKVCVETVESGAMTKDLAGCIHGLSNVKLNEHFLNTTDFLDTIKSNLDRALGRQ