Reaction Details
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Target
Bromodomain-containing protein 3 [24-144,306-416]
Ligand
BDBM205431
Substrate
n/a
Meas. Tech.
Bromodomains Assay for DiscoveRx Gene Symbol
Ki
0.11±0.0 nM
Citation
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More Info.:
Target
Name:
Bromodomain-containing protein 3 [24-144,306-416]
Synonyms:
BET bromodomain 3(1,2) (BRD3(1,2)) | BRD3 | BRD3_HUMAN | KIAA0043 | RING3L
Type:
n/a
Mol. Mass.:
27406.43
Organism:
Homo sapiens (Human)
Description:
Q15059 (BRD3, 24-144) and 306-416)
Residue:
232
Sequence:
PEVSNPSKPGRKTNQLQYMQNVVVKTLWKHQFAWPFYQPVDAIKLNLPDYHKIIKNPMDMGTIKKRLENNYYWSASECMQDFNTMFTNCYIYNKPTDDIVLMAQALEKIFLQKVAQMPQEEGKLSEHLRYCDSILREMLSKKHAAYAWPFYKPVDAEALELHDYHDIIKHPMDLSTVKRKMDGREYPDAQGFAADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKMP