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Target
Bromodomain-containing protein 4 [44-168,333-460]
Ligand
BDBM205431
Substrate
n/a
Meas. Tech.
BROMOscan Assay
Kd
0.0047±0.0 nM
Citation
Tanaka, M; Roberts, JM; Seo, HS; Souza, A; Paulk, J; Scott, TG; DeAngelo, SL; Dhe-Paganon, S; Bradner, JE Design and characterization of bivalent BET inhibitors. Nat Chem Biol 12:1089-1096 (2016) [PubMed] Article
More Info.:
Target
Name:
Bromodomain-containing protein 4 [44-168,333-460]
Synonyms:
BET bromodomain 4(1,2) (BRD4(1,2)) | BRD4 | BRD4_HUMAN | HUNK1
Type:
n/a
Mol. Mass.:
29666.85
Organism:
Homo sapiens (Human)
Description:
O60885 (BRD4, 44-168 and 333-460)
Residue:
253
Sequence:
NPPPPETSNPNKPKRQTNQLQYLLRVVLKTLWKHQFAWPFQQPVDAVKLNLPDYYKIIKTPMDMGTIKKRLENNYYWNAQECIQDFNTMFTNCYIYNKPGDDIVLMAEALEKLFLQKINELPTEEKDVPDSQQHPAPEKSSKVSEQLKCCSGILKEMFAKKHAAYAWPFYKPVDVEALGLHDYCDIIKHPMDMSTIKSKLEAREYRDAQEFGADVRLMFSNCYKYNPPDHEVVAMARKLQDVFEMRFAKMPDE