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Target
Bromodomain testis-specific protein [21-137,251-382]
Ligand
BDBM205431
Substrate
n/a
Meas. Tech.
BROMOscan Assay
Kd
0.039±0.0 nM
Citation
Tanaka, M; Roberts, JM; Seo, HS; Souza, A; Paulk, J; Scott, TG; DeAngelo, SL; Dhe-Paganon, S; Bradner, JE Design and characterization of bivalent BET inhibitors. Nat Chem Biol 12:1089-1096 (2016) [PubMed] Article
More Info.:
Target
Name:
Bromodomain testis-specific protein [21-137,251-382]
Synonyms:
BRDT | BRDT_HUMAN | Bromodomain testis (1, 2) (BRDT(1,2))
Type:
n/a
Mol. Mass.:
29512.81
Organism:
Homo sapiens (Human)
Description:
Q58F21 (BRDT, 21-137 and 251-382)
Residue:
249
Sequence:
NTKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEKNVLPDSQQQYNVVKTVKVTEQLRHCSEILKEMLAKKHFSYAWPFYNPVDVNALGLHNYYDVVKNPMDLGTIKEKMDNQEYKDAYKFAADVRLMFMNCYKYNPPDHEVVTMARMLQDVFETHFSKIPIEPVE