Reaction Details
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Target
Serine/threonine-protein kinase PAK 1 [249-545,K299R]
Ligand
BDBM50112347
Substrate
n/a
Meas. Tech.
Z'-LYTEBiochemical Assay
IC50
7.7±0.0 nM
Citation
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More Info.:
Target
Name:
Serine/threonine-protein kinase PAK 1 [249-545,K299R]
Synonyms:
PAK1 | PAK1_HUMAN | p21-Activated kinase 1 (PAK1)
Type:
Enzyme
Mol. Mass.:
33244.90
Organism:
Homo sapiens (Human)
Description:
Human PAK1 truncation (249-545 aa) with K299R mutation
Residue:
297
Sequence:
SDEEILEKLRSIVSVGDPKKKYTRFEKIGQGASGTVYTAMDVATGQEVAIRQMNLQQQPKKELIINEILVMRENKNPNIVNYLDSYLVGDELWVVMEYLAGGSLTDVVTETCMDEGQIAAVCRECLQALEFLHSNQVIHRDIKSDNILLGMDGSVKLTDFGFCAQITPEQSKRSTMVGTPYWMAPEVVTRKAYGPKVDIWSLGIMAIEMIEGEPPYLNENPLRALYLIATNGTPELQNPEKLSAIFRDFLNRCLEMDVEKRGSAKELLQHQFLKIAKPLSSLTPLIAAAKEATKNNH