Reaction Details Report a problem with these data
Target
Tyrosine-protein kinase SYK [360-635]
Ligand
BDBM227529
Substrate
n/a
Meas. Tech.
SYK Kinase Assay
Temperature
303.15±n/a K
IC50
2±n/a nM
Comments
extracted
Citation
Hermann, JC; Kennedy-Smith, J; Lucas, MC; Padilla, F; Schoenfeld, RC; Wovkulich, PM Pyrrolo[2,3-B]pyrazines as SYK inhibitors US Patent US9334278 Publication Date 5/10/2016
More Info.:
Target
Name:
Tyrosine-protein kinase SYK [360-635]
Synonyms:
KSYK_HUMAN | SYK | SYK RPA purified, truncated construct of Spleen Tyrosine Kinase (aa 360-635) | Tyrosine-protein kinase SYK | recombinant human SYK(aa 360-635)
Type:
n/a
Mol. Mass.:
31987.15
Organism:
Homo sapiens (Human)
Description:
Human MetAP2 protein from a culture superatant of insect cells (sf9) infected with MetAP2 recombinant baculovirus
Residue:
276
Sequence:
PKEVYLDRKLLTLEDKELGSGNFGTVKKGYYQMKKVVKTVAVKILKNEANDPALKDELLAEANVMQQLDNPYIVRMIGICEAESWMLVMEMAELGPLNKYLQQNRHVKDKNIIELVHQVSMGMKYLEESNFVHRDLAARNVLLVTQHYAKISDFGLSKALRADENYYKAQTHGKWPVKWYAPECINYYKFSSKSDVWSFGVLMWEAFSYGQKPYRGMKGSEVTAMLEKGERMGCPAGCPREMYDLMNLCWTYDVENRPGFAAVELRLRNYYYDVVN