Reaction Details
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Target
Thyroid hormone receptor alpha
Ligand
BDBM86689
Substrate
n/a
Ki
1250±n/a nM
Citation
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More Info.:
Target
Name:
Thyroid hormone receptor alpha
Synonyms:
C-erba-alpha | Nr1a1 | THA_RAT | Thra | Thyroid hormone receptor alpha | thyroid alpha
Type:
Enzyme Catalytic Domain
Mol. Mass.:
55077.31
Organism:
RAT
Description:
thyroid alpha 0 RAT::P63059
Residue:
492
Sequence:
MEQKPSKVECGSDPEENSARSPDGKRKRKNGQCPLKSSMSGYIPSYLDKDEQCVVCGDKATGYHYRCITCEGCKGFFRRTIQKNLHPTYSCKYDSCCVIDKITRNQCQLCRFKKCIAVGMAMDLVLDDSKRVAKRKLIEQNRERRRKEEMIRSLQQRPEPTPEEWDLIHVATEAHRSTNAQGSHWKQRRKFLPDDIGQSPIVSMPDGDKVDLEAFSEFTKIITPAITRVVDFAKKLPMFSELPCEDQIILLKGCCMEIMSLRAAVRYDPESDTLTLSGEMAVKREQLKNGGLGVVSDAIFELGKSLSAFNLDDTEVALLQAVLLMSTDRSGLLCVDKIEKSQEAYLLAFEHYVNHRKHNIPHFWPKLLMKEREVQSSILYKGAAAEGRPGGSLGVHPEGQQLLGMHVVQGPQVRQLEQQFGEAGSLRGPVLQHQSPKSPQQRLLELLHRSGILHSRAVCGEDDSSEASSLSSSSSDEDTEVFEDLAGKAASP