Reaction Details
Report a problem with these data
![](/images/Email.png)
Target
Protein farnesyltransferase alpha subunit/subunit beta
Ligand
BDBM238357
Substrate
n/a
Meas. Tech.
T. brucei FTase Assay
IC50
32000±5000 nM
Citation
More Info.:
Target
Name:
Protein farnesyltransferase alpha subunit/subunit beta
Synonyms:
Farnesyltransferase (FTase)
Type:
Enzyme
Mol. Mass.:
n/a
Description:
T. brucei FTase
Components:
This complex has 2 components.
Component 1
Name:
Protein farnesyltransferase alpha subunit
Synonyms:
Protein farnesyltransferase subunit alpha
Type:
Protein
Mol. Mass.:
70116.60
Organism:
Trypanosoma brucei brucei
Description:
Q9NC77
Residue:
612
Sequence:
MNKSAVRSEESRQSSSLPSTYSSSSLNSEDERLALLSDINALQALFPGVTPKEETPLIKHPNMTPAVFSKKFDYVMGIYRAVGVTFKGTRVGPSTPQWLLLTSFVIQQNASHYSAWKDRRDVFLQPSRLVTSTRDAFMAENGQQCCGDKTDSLAKVSQEWLPAQCDVQGPTGECSVWRAIRWELKAMERFALMNPKNFQVWHHRREMLREALMHANPVVTGSRSAFDGYLLTCHNMQFSDIDERVFCDAALDDDGKNYHAWLYRSWFVHSFPFLLHPPSWDSLLGGDQGTEDKHSELRAAPFRSFTVEEDWLHKCLQPIIPECPLSDELTSTAKRILHDCMNNSAWCHRFYVFEHDLIVPLIRVIPPQQTEEAKLILKRLCECEMFYALQWCAYEPCNESAFVHARCVAVLHQAVAIHLCLSSHGDAPHVFLRGDETIQVAGSSSLRHINLRDKLRWGAFLETFRLLLCQVNVLSDVITPRAEEFRSGGEGRDNATISVIHKRRSQFLLDNTHQVYTARYRCLFTILEYMWRCYFTVSDRANVAAALPPEVYAGGDAEAAALAQQQSDDCVKFFLEAELQALRLARRLVVEDDIRRKYWKHEMNIVMNRDYV
Component 2
Name:
Protein farnesyltransferase subunit beta
Synonyms:
n/a
Type:
Protein
Mol. Mass.:
65426.56
Organism:
Trypanosoma brucei brucei
Description:
Q9NC76
Residue:
585
Sequence:
MSFVPPPASSTTHAQREVELTLLRFLEKYRPEVCDLWGTHSDIHLHADSNEKEEEMCTIDNEEGIVHSLNRESHEKYLKSRLVKLPEYAQRLYNAQPWMVYWTLQAAEMLGITEKLYEQISQDALGEFILSCLQEQPVEDEQKGCWGSEEGGKHGKGSMPQQCGNVYDFLRRCDADHTCAIGFSGGNYGQIPHLATSYAGVCSLCILGCPEYLQALPRSAIKRWLLSLRCADGSFRMHIGGEADIRASYCVAVITTLLQLQDVDVRSGDILREQEAQFVASCQTHEGGFACGRFASEAHGAYTQCGLAALILMKRPELCNYTALRGWLAARQLRFEGGFNGRTNKLVDSCYAHWVGASHVLLRVGESLAKITTCGETKRSLTSREMLLLDHAQLVDISNLHPESFEAWSQHEEEKQERASRVEAYLSATPLAASWSSSGVPNVLDDDAGDFYFNQRRLQLYILACCQNREEGGLMDKPNYPNDFYHTCYSLSGMSSAQNLQGMQVNRDGRDLSGNSFYAAALSRGYIPGRRDSYGIVLPSDERSGVSSELHLSKNCLRPTNPIFNINQSKVLFALRTWGAKTFMC