Reaction Details Report a problem with these data
Target
Serine/threonine-protein kinase PLK4 [1-391]
Ligand
BDBM375451
Substrate
n/a
Meas. Tech.
Inhibition Assay
IC50
<100±n/a nM
Citation
Sampson, PB; Liu, Y; Li, S; Forrest, BT; Pauls, HW; Edwards, LG; Feher, M; Patel, NK; Laufer, R Kinase inhibitors and method of treating cancer US Patent US10358436 Publication Date 7/23/2019
More Info.:
Target
Name:
Serine/threonine-protein kinase PLK4 [1-391]
Synonyms:
PLK4 | PLK4_HUMAN | SAK | STK18 | Serine/threonine-protein kinase PLK4
Type:
Protein
Mol. Mass.:
43940.49
Organism:
Homo sapiens (Human)
Description:
aa 1-391
Residue:
391
Sequence:
MATCIGEKIEDFKVGNLLGKGSFAGVYRAESIHTGLEVAIKMIDKKAMYKAGMVQRVQNEVKIHCQLKHPSILELYNYFEDSNYVYLVLEMCHNGEMNRYLKNRVKPFSENEARHFMHQIITGMLYLHSHGILHRDLTLSNLLLTRNMNIKIADFGLATQLKMPHEKHYTLCGTPNYISPEIATRSAHGLESDVWSLGCMFYTLLIGRPPFDTDTVKNTLNKVVLADYEMPSFLSIEAKDLIHQLLRRNPADRLSLSSVLDHPFMSRNSSTKSKDLGTVEDSIDSGHATISTAITASSSTSISGSLFDKRRLLIGQPLPNKMTVFPKNKSSTDFSSSGDGNSFYTQWGNQETSNSGRGRVIQDAEERPHSRYLRRAYSSDRSGTSNSQSQA