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Target
Alpha-synuclein
Ligand
BDBM491853
Substrate
n/a
Meas. Tech.
In-Vitro Fluorescence Polarization Assay
IC50
1200±n/a nM
Citation
Wrasidlo, W; Stocking, EM; Hall, A; Maccoss, M Bis-heteroaryl derivatives as modulators of protein aggregation US Patent US10975066 Publication Date 4/13/2021
More Info.:
Target
Name:
Alpha-synuclein
Synonyms:
NACP | PARK1 | SNCA | SYUA_HUMAN
Type:
Protein
Mol. Mass.:
14451.42
Organism:
Homo sapiens (Human)
Description:
P37840
Residue:
140
Sequence:
MDVFMKGLSKAKEGVVAAAEKTKQGVAEAAGKTKEGVLYVGSKTKEGVVHGVATVAEKTKEQVTNVGGAVVTGVTAVAQKTVEGAGSIAAATGFVKKDQLGKNEEGAPQEGILEDMPVDPDNEAYEMPSEEGYQDYEPEA