Reaction Details
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Target
RAF proto-oncogene serine/threonine-protein kinase [1-324]
Ligand
BDBM202717
Substrate
n/a
Meas. Tech.
In Vitro Raf Activity
IC50
0.508±n/a nM
Citation
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More Info.:
Target
Name:
RAF proto-oncogene serine/threonine-protein kinase [1-324]
Synonyms:
C-Raf TR | P04049 (aa 1-324) | RAF | RAF proto-oncogene serine/threonine-protein kinase (aa 1-324) | RAF1 | RAF1_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42815.85
Organism:
Homo sapiens (Human)
Description:
P04049 (aa 1-324)
Residue:
384
Sequence:
MEHIQGAWKTISNGFGFKDAVFDGSSCISPTIVQQFGYQRRASDDGKLTDPSKTSNTIRVFLPNKQRTVVNVRNGMSLHDCLMKALKVRGLQPECCAVFRLLHEHKGKKARLDWNTDAASLIGEELQVDFLDHVPLTTHNFARKTFLKLAFCDICQKFLLNGFRCQTCGYKFHEHCSTKVPTMCVDWSNIRQLLLFPNSTIGDSGVPALPSLTMRRMRESVSRMPVSSQHRYSTPHAFTFNTSSPSSEGSLSQRQRSTSTPNVHMVSTTLPVDSRMIEDAIRSHSESASPSALSSSPNNLSPTGWSQPKTPVPAQRERAPVSGTQEKNKIRPRGQRDSSYYWEIEASEVMLSTRIGSGSFGTVYKGKWHGDVAVKILKVVDPTP