Reaction Details
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Target
Estrogen receptor [D538G]
Ligand
BDBM263664
Substrate
n/a
Meas. Tech.
Estrogen Receptor Coactivator Assay
pH
7.4±n/a
Temperature
298.15±n/a K
IC50
32.0±n/a nM
Comments
extracted
Citation
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More Info.:
Target
Name:
Estrogen receptor [D538G]
Synonyms:
ESR | ESR1 | ESR1_HUMAN | Estrogen receptor alpha D538G | NR3A1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
66173.42
Organism:
Homo sapiens (Human)
Description:
P03372[D538G]
Residue:
595
Sequence:
MTMTLHTKASGMALLHQIQGNELEPLNRPQLKIPLERPLGEVYLDSSKPAVYNYPEGAAYEFNAAAAANAQVYGQTGLPYGPGSEAAAFGSNGLGGFPPLNSVSPSPLMLLHPPPQLSPFLQPHGQQVPYYLENEPSGYTVREAGPPAFYRPNSDNRRQGGRERLASTNDKGSMAMESAKETRYCAVCNDYASGYHYGVWSCEGCKAFFKRSIQGHNDYMCPATNQCTIDKNRRKSCQACRLRKCYEVGMMKGGIRKDRRGGRMLKHKRQRDDGEGRGEVGSAGDMRAANLWPSPLMIKRSKKNSLALSLTADQMVSALLDAEPPILYSEYDPTRPFSEASMMGLLTNLADRELVHMINWAKRVPGFVDLTLHDQVHLLECAWLEILMIGLVWRSMEHPGKLLFAPNLLLDRNQGKCVEGMVEIFDMLLATSSRFRMMNLQGEEFVCLKSIILLNSGVYTFLSSTLKSLEEKDHIHRVLDKITDTLIHLMAKAGLTLQQQHQRLAQLLLILSHIRHMSNKGMEHLYSMKCKNVVPLYGLLLEMLDAHRLHAPTSRGGASVEETDQSHLATAGSTSSHSLQKYYITGEAEGFPATV