Reaction Details Report a problem with these data
Target
Outer capsid protein sigma-1
Ligand
BDBM82273
Substrate
n/a
Ki
158.48±n/a nM
Comments
PDSP_1621
Citation
Hegde, SS; Bonhaus, DW; Johnson, LG; Leung, E; Clark, RD; Eglen, RM RS 39604: a potent, selective and orally active 5-HT4 receptor antagonist. Br J Pharmacol 115:1087-95 (1995) [PubMed] Article
More Info.:
Target
Name:
Outer capsid protein sigma-1
Synonyms:
Outer capsid protein sigma-1 | S1 | SIGM1_REOVD | Sigma-1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
49088.08
Organism:
Mammalian orthoreovirus 3 Dearing
Description:
Sigma-1 0 0::P03528
Residue:
455
Sequence:
MDPRLREEVVRLIIALTSDNGASLSKGLESRVSALEKTSQIHSDTILRITQGLDDANKRIIALEQSRDDLVASVSDAQLAISRLESSIGALQTVVNGLDSSVTQLGARVGQLETGLAELRVDHDNLVARVDTAERNIGSLTTELSTLTLRVTSIQADFESRISTLERTAVTSAGAPLSIRNNRMTMGLNDGLTLSGNNLAIRLPGNTGLNIQNGGLQFRFNTDQFQIVNNNLTLKTTVFDSINSRIGATEQSYVASAVTPLRLNSSTKVLDMLIDSSTLEINSSGQLTVRSTSPNLRYPIADVSGGIGMSPNYRFRQSMWIGIVSYSGSGLNWRVQVNSDIFIVDDYIHICLPAFDGFSIADGGDLSLNFVTGLLPPLLTGDTEPAFHNDVVTYGAQTVAIGLSSGGAPQYMSKNLWVEQWQDGVLRLRVEGGGSITHSNSKWPAMTVSYPRSFT