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Target
5-hydroxytryptamine receptor 7
Ligand
BDBM50130269
Substrate
n/a
Ki
10±n/a nM
Comments
PDSP_1095
Citation
 Boess, FG; Martin, IL Molecular biology of 5-HT receptors. Neuropharmacology 33:275-317 (1994) [PubMed]  Article
Target
Name:
5-hydroxytryptamine receptor 7
Synonyms:
5-HT-7 | 5-HT-X | 5-HT7 | 5-hydroxytryptamine receptor 7 | 5-hydroxytryptamine receptor 7 (5HT7) | 5HT7 | 5HT7R_MOUSE | Htr7 | Serotonin 7 (5-HT7) receptor
Type:
Enzyme
Mol. Mass.:
49932.71
Organism:
Mus musculus (Mouse)
Description:
P32304
Residue:
448
Sequence:
MMDVNSSGRPDLYGHLRSLILPEVGRRLQDLSPDGGAHSVVSSWMPHLLSGFPEVTASPAPTWDAPPDNVSGCGEQINYGRVEKVVIGSILTLITLLTIAGNCLVVISVCFVKKLRQPSNYLIVSLALADLSVAVAVMPFVSVTDLIGGKWIFGHFFCNVFIAMDVMCCTASIMTLCVISIDRYLGITRPLTYPVRQNGKCMAKMILSVWLLSASITLPPLFGWAQNVNDDKVCLISQDFGYTIYSTAVAFYIPMSVMLFMYYQIYKAARKSAAKHKFSGFPRVQPESVISLNGVVKLQKEVEECANLSRLLKHERKNISIFKREQKAATTLGIIVGAFTVCWLPFFLLSTARPFICGTSCSCIPLWVERTCLWLGYANSLINPFIYAFFNRDLRTTYRSLLQCQYRNINRKLSAAGMHEALKLAERPERSEFVLQNCDHCGKKGHDT
  
Inhibitor
Name:
BDBM50130269
Synonyms:
(6aR,9R)-5-Bromo-7-methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid diethylamide | 5-Bromo-7-methyl-4,6,6a,7,8,9-hexahydro-indolo[4,3-fg]quinoline-9-carboxylic acid diethylamide | CHEMBL274384 | LSD,2-Bromo
Type:
Small organic molecule
Emp. Form.:
C20H24BrN3O
Mol. Mass.:
402.328
SMILES:
CCN(CC)C(=O)[C@H]1CN(C)[C@@H]2Cc3c(Br)[nH]c4cccc(C2=C1)c34 |c:23|
Structure:
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